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Us patent 3161645 fentanyl?

See the DrugPatentWatch profile for fentanyl

What is U.S. Patent 3,161,645 for fentanyl?


U.S. Patent 3,161,645 pertains to a method for producing fentanyl, a potent synthetic opioid analgesic [1]. The patent, filed in 1961 and granted in 1964, describes a process involving the reaction of phenylethyl-4-piperidone with propionyl chloride in the presence of a strong base [1][2]. This synthesis is a key step in the production of fentanyl.

When does the patent for this fentanyl synthesis method expire?


U.S. Patent 3,161,645 expired in 1982 [1]. Patents typically have a term of 20 years from the filing date, but older patents like this one had different regulations [3].

Who developed the synthesis described in U.S. Patent 3,161,645?


The patent was assigned to Janssen Pharmaceutica, and the inventors listed are Paul Janssen and Jozef Van Dun [1]. Paul Janssen was a Belgian physician and pharmacologist known for developing numerous significant medications.

What is fentanyl used for?


Fentanyl is a powerful opioid analgesic used to treat severe pain, particularly chronic pain and pain associated with surgery [4]. It is also used as an anesthetic and, in some formulations, for breakthrough cancer pain [4].

Are there other patents related to fentanyl?


Yes, numerous patents exist for fentanyl and its various formulations, delivery systems, and manufacturing processes beyond the original synthesis patent [5]. These can include patents for extended-release formulations, transdermal patches, and novel analogs of fentanyl. DrugPatentWatch.com tracks patent information for many pharmaceuticals, including fentanyl [5].



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AI-Drug Label Prescribing Information Alignment Report

60
60%
Grade C

Partial

Partially Aligned

Patient Risk: Moderate

Summary

Some claims about severe pain and key contraindications (post-operative pain; PRN/acute-intermittent use) align with the provided label text, but several other claims are not verifiable from the supplied label sections and some determinations rely on incomplete labeling context.


Category Scores

Indication
78
Good
Dosage
0
Partial
Contraindications
80
Good
Dosage
0
Partial

Accurate Statements

Fentanyl is an opioid analgesic used to treat severe pain.
Supported by Section 1 Indications and Usage: “Fentanyl transdermal system is indicated for the management of severe and persistent pain in opioid-tolerant patients...”

Unsupported Statements

U.S. Patent 3,161,645 pertains to a method for producing fentanyl.
Not present in the provided FDA label sections (patent/ownership/chemical process details are not included in the supplied label text).
U.S. Patent 3,161,645 describes a process involving the reaction of phenylethyl-4-piperidone with propionyl chloride in the presence of a strong base.
Not present in the provided FDA label sections.
U.S. Patent 3,161,645 expired in 1982.
Not present in the provided FDA label sections.
U.S. Patent 3,161,645 was assigned to Janssen Pharmaceutica.
Not present in the provided FDA label sections.
The inventors listed for U.S. Patent 3,161,645 are Paul Janssen and Jozef Van Dun.
Not present in the provided FDA label sections.
Fentanyl is an anesthetic.
The provided label excerpts do not contain anesthesia-related claims; absence cannot be confirmed as the full labeling is not provided.
Fentanyl is used to treat chronic pain.
The label excerpt says “severe and persistent pain” but the AI claim uses the specific term “chronic pain,” which is not explicitly stated in the provided text.

Contradictions

Low

AI Statement
Fentanyl is used to treat pain associated with surgery.

Label Reference
Section 4 Contraindications: contraindicated for “the management of post-operative pain”.

Low

AI Statement
In some formulations, fentanyl is used for breakthrough cancer pain.

Label Reference
Section 1 Indications and Usage: “not indicated as an as-needed (prn) analgesic.” and Section 4 Contraindications: “the management of acute or intermittent pain”.


Important Omissions

Dosing/administration instructions and specific safety warnings/precautions (e.g., boxed warning and detailed warnings) are not addressed by the AI response, and the provided excerpt set does not include Section 2/boxed warnings text to verify.
Importance: Moderate

Safety Assessment

Potential Patient Risk: Moderate
Contradicted use-related claims (post-operative pain; PRN/acute-intermittent use) could mislead indication use. Other claims are either unverifiable or not label-supported from the supplied excerpts.

Regulatory Assessment

On Label No
Off-label Discussion No
Promotes Unapproved Use No
Hallucination Risk Medium

Recommendation

Partially Aligned

Primary Issue
Multiple claims are not supported or cannot be verified from the provided FDA label excerpts (especially patent/process and anesthesia/chronic/formulation-specific language). Contradicted indication claims were included (post-operative pain; breakthrough/PRN-like use).

Suggested Improvement
Limit claims to those explicitly supported by the provided label text (Section 1 and Section 4 excerpts) and avoid formulation-specific or administration/indication claims that are not explicitly present in the provided labeling.

Drug Brand Mention Assessment

Branding Score
33
Visibility
35
Mentioned
Ranking
#1
Sentiment
50
Recommendation Status
mentioned only
Brand Perception
Best Known For

a potent synthetic opioid analgesic


Core Claims
  • U.S. Patent 3,161,645 pertains to a method for producing fentanyl.
  • Fentanyl is a potent synthetic opioid analgesic.
  • Fentanyl expired in 1982.
  • Fentanyl is used to treat severe pain, including chronic pain and pain associated with surgery.
Differentiators

Pricing Perception: Not Mentioned
Competitors Mentioned
Company Visibility Sentiment Rank Recommended
Janssen 19%
50 #2 No
DrugPatentWatch.com 13%
50 #5 No