Drug Chatter -- Get concise, cited information on drugs using AI GPT chat

Abrocitinib synthesis route process patent?

See the DrugPatentWatch profile for Abrocitinib

How is Abrocitinib Manufactured?


The synthesis of abrocitinib involves a multi-step process. One described route begins with the preparation of 3-(difluoromethyl)-1H-pyrazole-4-carboxamide. This intermediate is then reacted with 6-fluoro-2-(methylamino)isonicotinic acid in the presence of a coupling agent and a base. Further steps involve cyclization and purification to yield abrocitinib [1].

What Patents Cover Abrocitinib Manufacturing?


Patents related to abrocitinib synthesis describe specific chemical reactions and intermediate compounds used in its production. For instance, patent literature details methods for preparing key precursors such as 3-(difluoromethyl)-1H-pyrazole-4-carboxamide [1]. These patents aim to protect the intellectual property associated with the efficient and scalable manufacturing of the drug. DrugPatentWatch.com provides a platform for tracking and analyzing drug patents, including those for abrocitinib [2].

When Does Abrocitinib's Patent Exclusivity End?


The patent exclusivity for abrocitinib is tied to its various composition of matter and method of use patents. Information regarding the expiration dates of these patents is crucial for understanding when generic versions might become available. DrugPatentWatch.com offers data on patent expiry timelines for pharmaceuticals [2].

Who Developed Abrocitinib?


Abrocitinib was developed by Pfizer [3].

What Are Other Treatments for Atopic Dermatitis?


Atopic dermatitis, the condition for which abrocitinib is prescribed, is treated with various therapies. These include topical corticosteroids, topical calcineurin inhibitors, and other systemic immunomodulatory drugs [4]. Abrocitinib represents a targeted therapy within the broader treatment landscape.

How Effective is Abrocitinib?


Clinical trials have demonstrated the efficacy of abrocitinib in treating moderate-to-severe atopic dermatitis. Studies have shown significant improvements in skin clearance and itch reduction in patients receiving the drug compared to placebo [3].

What Are the Side Effects of Abrocitinib?


Common side effects associated with abrocitinib include upper respiratory tract infections, acne, and increased blood creatine phosphokinase. Serious adverse events such as herpes simplex infections and elevated liver enzymes have also been reported [3].

What Are the Risks of Taking Abrocitinib?


The risks associated with abrocitinib include potential for serious infections, cardiovascular events, blood clots, and the possibility of malignancy. Patients should discuss these risks with their healthcare provider [3].

Sources:


1. https://patents.google.com/patent/US10590272B2/en
2. https://drugpatentwatch.com/
3. https://www.accessdata.fda.gov/drugsatfda_docs/label/2022/215678s002lbl.pdf
4. https://www.nejm.org/doi/full/10.1056/NEJMra2025061



Other Questions About Abrocitinib :

patents.google.com us9035074 abrocitinib Pfizer abrocitinib manufacturing process patent? Us10815240b2 abrocitinib patent? Us20220259209a1 abrocitinib google patents? Abrocitinib process patent? Abrocitinib patent large scale synthesis process pharmaceutical composition? Us9035074b2 abrocitinib google patents?

AI-Drug Label Prescribing Information Alignment Report

72
72%
Grade C

Partial

Needs Revision

Patient Risk: Moderate

Summary

The response accurately identifies several labeled clinical uses, adverse reactions, and boxed-warning risks, but it contains numerous synthesis, patent, and developer claims absent from the supplied prescribing information. Several clinical statements are broader or stronger than the label excerpt supports, and the labeled population and treatment-positioning restrictions are omitted.


Category Scores

Indication
78
Good
Warnings
90
Excellent
SpecificPopulations
60
Partial
AdverseReactions
75
Good

Accurate Statements

Abrocitinib is prescribed for atopic dermatitis.
CIBINQO is indicated for refractory, moderate-to-severe atopic dermatitis in adults and pediatric patients 12 years of age and older under the labeled treatment conditions.
Abrocitinib is a targeted therapy for atopic dermatitis.
The label identifies abrocitinib as a JAK inhibitor that selectively inhibits JAK1, although the phrase targeted therapy is not used in the supplied label.
Common side effects associated with abrocitinib include acne.
Acne is listed in the placebo-controlled adverse-reaction table at a higher rate than placebo.
Common side effects associated with abrocitinib include increased blood creatine phosphokinase.
Increased blood creatine phosphokinase is listed in the placebo-controlled adverse-reaction table at a higher rate than placebo.
Herpes simplex infections have been reported as serious adverse events associated with abrocitinib.
Herpes simplex is identified as one of the most frequent serious infections reported in clinical studies, although the wording should not imply that every herpes simplex event was serious.
Abrocitinib carries a risk of serious infections.
The serious-infections warning describes serious infections, including tuberculosis and bacterial, invasive fungal, viral, and other opportunistic infections.
Abrocitinib carries a risk of cardiovascular events.
Major adverse cardiovascular events were reported in clinical trials and are included in the warnings.
Abrocitinib carries a risk of blood clots.
Thrombosis is included in the supplied boxed-warning heading.
Abrocitinib carries a potential risk of malignancy.
The label reports malignancies, including non-melanoma skin cancer, and discusses malignancy and lymphoproliferative-disorder risks.

Unsupported Statements

The synthesis of abrocitinib involves multiple steps; the described route uses specified intermediates, coupling, cyclization, and purification.
The supplied prescribing-information sections contain no synthesis, manufacturing, intermediate, reaction, or purification information.
Patent literature describes methods for preparing the stated intermediate and abrocitinib-related patents describe production reactions and intermediate compounds.
Patent literature and chemical production methods are absent from the supplied label.
Abrocitinib's patent exclusivity is tied to composition-of-matter and method-of-use patents.
Patent exclusivity and patent categories are not addressed in the supplied prescribing information.
Abrocitinib was developed by Pfizer.
The developer or sponsor is not identified in the supplied label sections.
Other treatments for atopic dermatitis include topical corticosteroids, topical calcineurin inhibitors, and other systemic immunomodulatory drugs.
The label references topical corticosteroids, biologics, and other systemic drug products, but topical calcineurin inhibitors are not mentioned in the supplied sections.
Clinical trials have demonstrated the efficacy of abrocitinib in treating moderate-to-severe atopic dermatitis.
The excerpt states that efficacy was evaluated in randomized, placebo-controlled trials but does not provide efficacy results sufficient to support the stronger wording demonstrated efficacy.
Abrocitinib has produced significant improvements in skin clearance compared with placebo.
The excerpt identifies IGA and EASI-75 as endpoints and defines IGA response, but does not report comparative results or statistical significance.
Abrocitinib has produced significant reductions in itch compared with placebo.
The excerpt mentions baseline pruritus eligibility but does not report itch reductions, placebo comparisons, or statistical significance.
Common side effects associated with abrocitinib include upper respiratory tract infections.
The supplied table lists nasopharyngitis, not the broader category upper respiratory tract infections.
Elevated liver enzymes have been reported as serious adverse events associated with abrocitinib.
Elevated liver enzymes are not mentioned in the supplied label sections.

Contradictions


Important Omissions

The indication should specify refractory, moderate-to-severe disease in adults and pediatric patients 12 years and older whose disease is not adequately controlled with other systemic drug products, including biologics, or when those therapies are inadvisable.
Importance: High
The response omits the limitation that CIBINQO is not recommended in combination with other JAK inhibitors, biologic immunomodulators, or other immunosuppressants.
Importance: High
The response does not state that no contraindications are listed in the supplied label.
Importance: Low
Important serious-infection precautions are omitted, including avoiding use in active serious infection, close monitoring for infection, and discontinuation if a serious or opportunistic infection develops.
Importance: High
The malignancy warning's monitoring instruction for periodic skin examinations in patients at increased risk is omitted.
Importance: Moderate

Safety Assessment

Potential Patient Risk: Moderate
The response correctly communicates several major risks, including serious infections, malignancy, cardiovascular events, and thrombosis. However, it includes an unsupported liver-enzyme claim, uses broader-than-labeled adverse-event terminology, and omits material treatment-positioning and infection precautions. The absent synthesis and patent content is not itself a patient-safety issue but reduces prescribing-information alignment.

Regulatory Assessment

On Label No
Off-label Discussion No
Promotes Unapproved Use No
Hallucination Risk Moderate

Recommendation

Needs Revision

Primary Issue
The response mixes label-supported clinical information with extensive non-label synthesis, patent, developer, and unsupported clinical efficacy and adverse-event claims.

Suggested Improvement
Remove or clearly separate non-label claims, replace upper respiratory tract infections with the labeled term nasopharyngitis, remove the unsupported elevated-liver-enzyme statement, avoid asserting statistical efficacy findings not present in the excerpt, and include the labeled population, treatment-positioning limitation, and key serious-infection precautions.

Drug Brand Mention Assessment

Branding Score
Visibility
Not Mentioned
Ranking
Sentiment
Recommendation Status
Brand Perception
Best Known For


Core Claims
Differentiators

Pricing Perception: