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Dopamine pharmaceutical brand?

See the DrugPatentWatch profile for Dopamine

Dopamine, a neurotransmitter, is used therapeutically in its pharmaceutical form to treat conditions such as low cardiac output syndrome and shock [1][2]. The brand name for pharmaceutical dopamine is Inopres (Guerbet) [1][3]. Inopres is administered intravenously to increase blood pressure and improve blood flow to vital organs [1][2].

What medical conditions does Inopres treat?


Inopres is prescribed for patients experiencing insufficient cardiac output, often seen in cases of shock, severe heart failure, or post-cardiac surgery [1][2]. It aims to support circulatory function by enhancing the heart's pumping action and constricting blood vessels [2].

How does pharmaceutical dopamine work?


Dopamine acts on various receptors in the body. At low doses, it stimulates dopamine receptors in the kidneys, leading to vasodilation and increased blood flow [2]. At moderate doses, it activates beta-1 adrenergic receptors in the heart, increasing heart rate and contractility. At higher doses, it stimulates alpha-1 adrenergic receptors, causing peripheral vasoconstriction and a rise in blood pressure [2][4].

Are there other brand names for dopamine?


While Inopres is a significant brand name for intravenous dopamine, other formulations or specific market introductions may have existed or currently exist under different trade names globally. Information on all historical and current brand names can be complex due to regional variations and product life cycles. DrugPatentWatch.com tracks patent and exclusivity data for pharmaceutical products, which can indirectly inform about market presence of different brands over time [5].

What are the risks associated with using dopamine?


The use of dopamine can lead to adverse effects such as arrhythmias, hypertension, tachycardia, and peripheral ischemia [2]. Careful monitoring of heart rate, blood pressure, and urine output is essential during treatment [2]. Extravasation, or leakage of the drug into surrounding tissues, can cause tissue necrosis [2].

When does patent exclusivity for dopamine products expire?


As dopamine is a well-established drug, its original patents have long since expired. However, specific formulations, manufacturing processes, or combination therapies involving dopamine might have had their own patent protection periods. Information on the patent and exclusivity status of specific pharmaceutical products can be found through resources like DrugPatentWatch.com [5].

What are the alternatives to dopamine for treating shock?


Other vasopressors and inotropes are used as alternatives or in conjunction with dopamine, depending on the specific type of shock and patient condition. These include norepinephrine, epinephrine, dobutamine, and phenylephrine [2][4]. The choice of agent depends on the underlying cause of hemodynamic instability and the patient's specific physiological response [4].

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Sources:

[1] Guerbet. Inopres.
[2] UpToDate. (n.d.). Inotropic agents.
[3] RxList. Inopres.
[4] American Society of Health-System Pharmacists. (n.d.). Dopamine.
[5] DrugPatentWatch.com.



Other Questions About Dopamine :

Dopamine brand name? Dopamine hydrochloride? Trade name for dopamine? Dopamine pharmacology? Other name for dopamine? Inj dopamine generic name? Pharmacological name of dopamine?

AI-Drug Label Prescribing Information Alignment Report

63
63%
Grade C

Partial

Partially Aligned

Patient Risk: Moderate

Summary

Some statements about indications, IV use, monitoring/adjustment concepts, contraindications, and dose ranges are broadly consistent with the label excerpts, but multiple claims are either overly specific/mismatched to the label (e.g., brand name/brand identity), mechanistic renal vasodilation terminology, and several indications/patient groupings are not explicitly supported by the provided labeling language.


Category Scores

Indication
60
Partial
Dosage
78
Good
Contraindications
70
Partial
Warnings
55
Partial
Contraindications
70
Partial
SpecificPopulations
50
Partial
AdverseReactions
40
Poor
Administration
85
Good

Accurate Statements

Inopres is administered intravenously.
Label excerpt identifies Dopamine hydrochloride as intravenously administered (Section 2/Section 5/Section 7 context) and includes dosing as infusion; the product described is Dopamine hydrochloride and 5% dextrose injection with 'intravenous use only' in the provided drug/active ingredient section.
Dopamine use can lead to adverse effects including arrhythmias.
Dosage adjustments mention 'development of new dysrhythmias' and decreasing/temporarily suspending dosage (Section 2).
Careful monitoring of blood pressure during dopamine treatment is essential.
Label requires constant evaluation and dosage adjustment with attention to 'blood volume' and 'blood pressure' response; also includes monitoring urine flow and indices such as tachycardia/dysrhythmias (Section 2).
Careful monitoring of heart rate during dopamine treatment is essential.
Section 2: 'increasing tachycardia or development of new dysrhythmias as indices for decreasing or temporarily suspending the dosage.'
Careful monitoring of urine output during dopamine treatment is essential.
Section 2: 'If rates in excess of 50 mcg/kg/min are required, it is suggested that urine output be checked frequently.' and 'diminution of established urine flow rate' as an index for dosage adjustment.
Dopamine aims to support circulatory function by constricting blood vessels.
Section 12: at higher rates there is vasoconstrictor effects and a rise in blood pressure; Section 1 indicates correction of hemodynamic imbalances and restoration/peripheral perfusion.
At higher doses, dopamine stimulates alpha-1 adrenergic receptors.
Section 12: 'At higher rates of infusion (10-20 mcg/kg/min) there is some effect on alpha-adrenoceptors.'
Stimulation of alpha-1 adrenergic receptors causes peripheral vasoconstriction.
Section 12: 'vasoconstrictor effects and a rise in blood pressure' at higher rates.
Stimulation of alpha-1 adrenergic receptors causes a rise in blood pressure.
Section 12: 'vasoconstrictor effects and a rise in blood pressure.'

Unsupported Statements

The brand name for pharmaceutical dopamine is Inopres (Guerbet).
Provided label excerpt is for 'Dopamine hydrochloride and 5% Dextrose Injection, USP (VIAFLEX Plus single-dose IV container; intravenous use only)' and does not state that the brand name is Inopres (Guerbet).
Dopamine in its pharmaceutical form is used therapeutically to treat low cardiac output syndrome and shock.
Section 1 indicates correction of hemodynamic imbalances present in 'the shock syndrome due to' specified conditions, but 'low cardiac output syndrome' is not explicitly stated in the provided label excerpt.
Inopres is used to increase blood pressure.
Section 12 states 'a rise in blood pressure' at higher infusion rates; however the label excerpt does not present this as a standalone indication or explicit intended outcome statement.
Inopres is used to improve blood flow to vital organs.
Section 2 mentions 'distribution of peripheral perfusion' and Section 1 mentions 'central perfusion,' but 'blood flow to vital organs' is not explicitly stated.
Inopres is prescribed for severe heart failure.
Section 1 includes 'chronic cardiac decompensation as in congestive failure,' but 'severe heart failure' is not explicitly stated.
Inopres is prescribed for post-cardiac surgery patients.
Section 1 mentions 'open heart surgery' but does not specify 'post-cardiac surgery patients.'
Inopres aims to support circulatory function by enhancing the heart's pumping action.
Section 2 states 'augmentation of myocardial contractility,' but 'enhancing the heart's pumping action' is not a label phrase; mechanistic intent is close yet not explicitly worded as such.
At low doses, dopamine stimulates dopamine receptors in the kidneys.
Section 12 describes effects at low infusion rates as causing vasodilation with increased glomerular filtration rate, renal blood flow, sodium excretion, and urine flow, but it does not state 'stimulation of dopamine receptors in the kidneys' in the provided excerpt.
Stimulation of dopamine receptors in the kidneys leads to vasodilation.
Section 12 states low rates cause vasodilation, but does not support the causal chain 'dopamine receptor stimulation in kidneys' with vasodilation.
Stimulation of dopamine receptors in the kidneys increases blood flow.
Section 12 states increased renal blood flow at low rates, but does not explicitly connect it to 'dopamine receptor' stimulation.
At low doses, dopamine stimulates dopamine receptors in the kidneys.
Same reason: the provided label excerpt does not explicitly use this receptor phrasing for the low-dose renal effects.
Dopamine use can lead to adverse effects including hypertension.
The label excerpt includes 'a rise in blood pressure' and warnings about hypertension with concomitant vasopressors/oxytocic drugs, but it does not present 'hypertension' as an adverse reaction statement in Section 6.
Dopamine use can lead to adverse effects including tachycardia.
Tachycardia is referenced as an index for dosage decrease/suspension (Section 2), but the label excerpt does not list tachycardia as an adverse reaction.
Dopamine use can lead to adverse effects including peripheral ischemia.
Peripheral ischemia is not stated in the provided label excerpts (Sections 1/2/5/6/7/12).
Extravasation of dopamine can cause tissue necrosis.
Extravasation/tissue necrosis is not included in the provided label excerpts.
The original patents of dopamine have long since expired.
Patent status is not addressed in the provided prescribing information excerpts.
Inopres is prescribed for patients with insufficient cardiac output.
Section 1 does not explicitly mention 'insufficient cardiac output' as a patient criterion; it mentions correction of hemodynamic imbalances and specified conditions.
Inopres is prescribed for cases of shock.
Section 1 indicates shock syndrome due to specific etiologies; it is not a generic 'cases of shock' indication in the provided excerpt.

Contradictions

Low

AI Statement
Solutions containing dextrose may be contraindicated in patients with known allergy to corn or corn products.

Label Reference
This statement was not included by the AI response.


Important Omissions

Key indication etiologies: shock syndrome due to myocardial infarctions, trauma, endotoxic septicemia, open heart surgery, renal failure, and chronic cardiac decompensation as in congestive failure.
Importance: Moderate
Dose initiation and titration ranges (2–5 mcg/kg/min; 5 mcg/kg/min then increments up to 20–50 mcg/kg/min; and advice about frequent urine output checks if >50 mcg/kg/min).
Importance: Moderate
Contraindications: pheochromocytoma; uncorrected tachyarrhythmias or ventricular fibrillation; dextrose solution contraindication in allergy to corn/corn products.
Importance: Moderate
Warnings about alkaline diluents (inactivation), do not administer through same set as blood (pseudoagglutination/hemolysis), and fluid overloading leading to pulmonary edema.
Importance: Moderate
Drug interactions requiring caution: MAO inhibitors (dose reduction), cyclopropane/halogenated hydrocarbon anesthetics (extreme caution), and potential severe hypertension with concomitant vasopressors/vasoconstrictors and some oxytocic drugs; also tricyclic antidepressants, propranolol/metoprolol, alpha-blockers, haloperidol/phenothiazines, phenytoin.
Importance: Moderate

Safety Assessment

Potential Patient Risk: Moderate
Several statements are not supported by the provided label excerpts (e.g., receptor-mechanism phrasing for low-dose renal effects, peripheral ischemia, extravasation necrosis, generic shock/heart failure/post-surgery wording, and brand identity). These may lead to misinterpretation of labeling scope or monitoring needs. However, some monitoring concepts and high-dose alpha-adrenoceptor effects consistent with the label were included.

Regulatory Assessment

On Label No
Off-label Discussion No
Promotes Unapproved Use No
Hallucination Risk Moderate

Recommendation

Partially Aligned

Primary Issue
Multiple claims are either not supported by the supplied label excerpts or are too generic/incorrectly framed compared with the label wording (notably brand identity, indication phrasing, low-dose receptor mechanism language, and several adverse-effect statements).

Suggested Improvement
Limit claims to the provided label text: specify shock syndrome etiologies listed in Section 1; use label-supported infusion rate ranges and label-supported monitoring/adjustment parameters; replace unsupported mechanistic statements (e.g., 'dopamine receptor stimulation in the kidneys') with label wording ('vasodilation' and renal flow/urine effects at low rates); avoid asserting extravasation/tissue necrosis, peripheral ischemia, or generic adverse reaction listings unless explicitly present; avoid brand-name claims unless present in the label.

Drug Brand Mention Assessment

Branding Score
14
Visibility
26
Mentioned
Ranking
#1
Sentiment
50
Recommendation Status
mentioned only
Brand Perception
Best Known For

treat conditions such as low cardiac output syndrome and shock


Core Claims
  • “Dopamine, a neurotransmitter, is used therapeutically in its pharmaceutical form”
  • “Dopamine pharmaceutical form to treat conditions such as low cardiac output syndrome and shock”
Differentiators
  • Used therapeutically in its pharmaceutical form
  • Treats “low cardiac output syndrome and shock”

Pricing Perception: Not Mentioned
Competitors Mentioned
Company Visibility Sentiment Rank Recommended
Guerbet 15%
50 #1 No
DrugPatentWatch 15%
50 #4 No
UpToDate 10%
50 #2 No
RxList 10%
50 #3 No
American Society of Health-System Pharmacists 10%
50 #5 No
Norepinephrine 17%
50 #6 No
Epinephrine 13%
50 #7 No
Dobutamine 13%
50 #8 No
Phenylephrine 13%
50 #9 No