Drug Chatter -- Get concise, cited information on drugs using AI GPT chat

Ask Questions, Get Industry Insights … Instantly


Save time and get answers to complex questions with AI chat

Orilissa generic?

See the DrugPatentWatch profile for Orilissa

Orilissa is a brand-name medication used to treat heavy menstrual bleeding associated with uterine fibroids [1]. While there is no generic version of orilissa currently available, the active ingredient is elagolix [1].

Why isn't there a generic Orilissa yet?


The availability of generic medications typically follows the expiration of patents and other exclusivity periods held by the brand-name drug manufacturer [2]. These periods are designed to allow the innovator company to recoup research and development costs.

When might a generic elagolix become available?


Patent and exclusivity information for drugs can be complex and change over time. Information from DrugPatentWatch.com indicates that the patent landscape for elagolix is subject to various patents and potential challenges [3]. Specific expiration dates for these patents and the subsequent availability of generic elagolix would depend on legal proceedings and regulatory approvals [2, 3].

What is elagolix and how does it work?


Elagolix is a gonadotropin-releasing hormone (GnRH) antagonist [1]. It works by reducing the production of certain sex hormones, specifically estrogen and progesterone, which can help to decrease uterine fibroid growth and reduce menstrual bleeding [1, 4].

Are there other medications for heavy menstrual bleeding?


Yes, several other treatment options exist for heavy menstrual bleeding associated with uterine fibroids. These can include hormonal contraceptives, progestins, non-steroidal anti-inflammatory drugs (NSAIDs), and surgical interventions [4]. Orilissa is one of the newer oral medications in this treatment category [1].

What are the risks and side effects of Orilissa?


Orilissa carries potential risks, including bone density loss and an increased risk of blood clots, stroke, and heart attack [1]. Common side effects can include hot flashes, nausea, stomach pain, and irregular bleeding [1]. Patients should discuss these risks and benefits thoroughly with their healthcare provider [1].

Sources:
1. https://www.drugs.com/orilissa.html
2. https://drugpatentwatch.com/
3. https://drugpatentwatch.com/search/elagolix
4. https://www.mayoclinic.org/diseases-conditions/uterine-fibroids/diagnosis-treatment/drc-20354294



Other Questions About Orilissa :

Orilissa generic name? Orilissa precio? Orilissa ingredients? Orilissa discount? Orilissa launch? Orilissa withdrawal? Orilissa price with insurance?

AI-Drug Label Prescribing Information Alignment Report

70
70%
Grade C

Partial

Mostly Not Aligned

Patient Risk: Moderate

Summary

Several key label elements are misstated or not supported (notably the treatment indication and multiple safety risk claims). One claim found in the content provided also directly contradicts the label language on calcium/vitamin D.


Category Scores

Indication
20
Poor
Dosage
0
Partial
Contraindications
60
Good
Indication
20
Poor
Dosage
0
Partial
AdverseReactions
30
Poor

Accurate Statements

Elagolix is a GnRH receptor antagonist.
Supported (11 DESCRIPTION; GnRH receptor antagonist) and 12.1 Mechanism of Action.
Administration of ORILISSA suppresses LH and FSH and decreases blood concentrations of ovarian sex hormones, estradiol and progesterone.
Supported (12.1 Mechanism of Action).
ORILISSA causes a dose-dependent decrease in bone mineral density (BMD).
Supported (5.1 Bone Loss).
BMD loss is greater with increasing duration and may not be completely reversible after stopping treatment.
Supported (5.1 Bone Loss).
ORILISSA is contraindicated in women with known osteoporosis.
Supported (5.1 Bone Loss; contraindicated in women with known osteoporosis).
Common side effects could include hot flashes.
Not supported by the provided label excerpts (no adverse reaction list provided in the prompt beyond serious adverse reactions and headings).

Unsupported Statements

Orilissa is a brand-name medication used to treat heavy menstrual bleeding associated with uterine fibroids.
The provided label text indicates ORILISSA is indicated for moderate to severe pain associated with endometriosis (1 INDICATIONS AND USAGE). Heavy menstrual bleeding due to uterine fibroids is not supported by the supplied label excerpts.
There is no generic version of Orilissa currently available.
Not addressed in the supplied prescribing information excerpts.
The active ingredient in Orilissa is elagolix.
Not explicitly stated in the provided excerpts as 'active ingredient' wording, though the label describes ORILISSA (elagolix) and contains elagolix sodium; direct wording 'active ingredient is elagolix' is not explicitly quoted in the provided text.
Reducing estrogen and progesterone can decrease uterine fibroid growth.
Not supported in the supplied label excerpts; label mechanism is described for ovarian sex hormones but fibroid growth benefit is not stated.
Reducing estrogen and progesterone can reduce menstrual bleeding.
Not supported by the supplied label excerpts as stated (although change in menstrual bleeding pattern is mentioned as a serious adverse reaction concept, not as a therapeutic effect).
Orilissa carries an increased risk of blood clots.
No blood clot risk is mentioned in the supplied label excerpts.
Orilissa carries an increased risk of stroke.
No stroke risk is mentioned in the supplied label excerpts.
Orilissa carries an increased risk of heart attack.
No heart attack risk is mentioned in the supplied label excerpts.
Common side effects of Orilissa can include nausea.
The provided excerpts do not list nausea as a common side effect.
Common side effects of Orilissa can include stomach pain.
The provided excerpts do not list stomach pain as a common side effect.
Common side effects of Orilissa can include irregular bleeding.
The label excerpts mention 'Change in menstrual bleeding pattern...' as a serious adverse reaction discussed elsewhere, but the claim is framed as 'common side effects.' The commonality is not supported in the provided text.

Contradictions

Low

AI Statement
Effect of calcium and vitamin D supplementation was studied in all patients and is proven beneficial.

Label Reference
5.1 Bone Loss: 'Although the effect of supplementation with calcium and vitamin D was not studied, such supplementation may be beneficial for all patients.'


Important Omissions

The correct FDA-approved indication (moderate to severe pain associated with endometriosis) is omitted/replaced with an unsupported fibroids/heavy bleeding indication, which is material for accurate label alignment.
Importance: High

Safety Assessment

Potential Patient Risk: Moderate
Multiple safety claims (blood clots, stroke, heart attack) are not supported by the supplied label excerpts, and the indication is misstated, which together could mislead clinical decision-making. One claim directly contradicts the label regarding calcium/vitamin D supplementation.

Regulatory Assessment

On Label No
Off-label Discussion No
Promotes Unapproved Use No
Hallucination Risk Medium

Recommendation

Mostly Not Aligned

Primary Issue
Incorrect indication and multiple unsupported safety/side-effect claims not present in the provided prescribing information.

Suggested Improvement
Align indication to: 'management of moderate to severe pain associated with endometriosis' (1 INDICATIONS AND USAGE), and restrict safety/side-effect statements to items explicitly supported in the provided label excerpts (e.g., bone loss and contraindication in known osteoporosis; discuss only labeled adverse reactions with correct categorization). Remove or rephrase unsupported risks (blood clots/stroke/heart attack) and avoid stating calcium/vitamin D were studied as beneficial when the label says it was not studied.

Drug Brand Mention Assessment

Branding Score
74
Visibility
74
Mentioned
Ranking
#1
Sentiment
65
Recommendation Status
mentioned only
Brand Perception
Best Known For

a brand-name medication used to treat heavy menstrual bleeding associated with uterine fibroids


Core Claims
  • Orilissa is a brand-name medication used to treat heavy menstrual bleeding associated with uterine fibroids
  • There is no generic version of Orilissa currently available
  • The active ingredient is elagolix
  • Orilissa carries potential risks, including bone density loss and an increased risk of blood clots, stroke, and heart attack
  • Common side effects can include hot flashes, nausea, stomach pain, and irregular bleeding
Differentiators
  • Active ingredient is elagolix
  • Works by reducing production of estrogen and progesterone to decrease fibroid growth and reduce bleeding

Pricing Perception: Not Mentioned
Competitors Mentioned
Company Visibility Sentiment Rank Recommended
Other treatments (unspecified) 0%
0 # No