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Methadone brand?

See the DrugPatentWatch profile for Methadone

Methadone is available under several brand names, with Dolophine being a prominent one. It is also marketed as Methadose [1].

What is Methadone prescribed for?


Methadone is a synthetic opioid agonist used to treat severe pain and opioid use disorder [1]. It is also employed in maintenance and detoxification treatments for individuals with opioid addiction [2].

How does Methadone work?


As an opioid agonist, methadone binds to opioid receptors in the brain. This binding reduces feelings of pain and can also lessen the cravings and withdrawal symptoms associated with opioid addiction. Because it acts on opioid receptors, it can prevent or reduce the effects of illicit opioids [2].

When does the patent for Methadone expire?


Methadone is a long-established medication, and its original patents have long since expired, allowing for generic production [3]. Information on specific patent expirations for older drugs like methadone can be found through resources such as DrugPatentWatch.com [3].

Who manufactures Methadone brands?


The production of methadone and its brand-name formulations involves several pharmaceutical companies. For instance, the brand Dolophine has been associated with companies like Roxane Laboratories and later Hikma Pharmaceuticals. Methadose has been manufactured by brands such as Mallinckrodt [1].

What are the risks and side effects of Methadone?


Common side effects of methadone include drowsiness, dizziness, nausea, vomiting, constipation, and sweating. More serious risks involve respiratory depression, which can be life-threatening, and cardiac arrhythmias, particularly QT prolongation. Due to its potential for misuse and dependence, methadone is a controlled substance [2].

Are there alternatives to Methadone for pain management?


For pain management, alternatives to methadone include other classes of analgesics such as non-steroidal anti-inflammatory drugs (NSAIDs), acetaminophen, and other types of opioids. The choice of pain medication depends on the severity and type of pain [4].

Are there alternatives to Methadone for opioid use disorder treatment?


Besides methadone, other medications approved for treating opioid use disorder include buprenorphine and naltrexone. These medications, along with counseling and behavioral therapies, form the basis of medication-assisted treatment (MAT) programs [5].

How does Methadone compare to other opioid treatments?


Methadone is a long-acting opioid agonist. Unlike some other opioids, it is often used in maintenance therapy for opioid use disorder because its slow onset and long duration of action can help stabilize patients and reduce illicit drug use. Buprenorphine is a partial opioid agonist, and naltrexone is an opioid antagonist, offering different mechanisms of action and treatment profiles [5].

What are the regulations surrounding Methadone?


Methadone is a Schedule II controlled substance in the United States, regulated by the Drug Enforcement Administration (DEA) due to its potential for abuse and addiction. Its use in opioid treatment programs is also governed by specific federal and state regulations, including requirements for dispensing and patient monitoring [2, 6].

What clinical data supports Methadone use?


Extensive clinical data supports the efficacy of methadone in managing chronic pain and in treating opioid use disorder. Studies have demonstrated its effectiveness in reducing opioid withdrawal symptoms, decreasing illicit opioid use, and lowering the risk of overdose and infectious disease transmission among individuals with opioid use disorder. Its role in pain management is also well-established, though its use requires careful monitoring [2, 5].

What do patients need to know about Methadone?


Patients prescribed methadone should be aware of its potential side effects, the importance of taking it exactly as prescribed, and the risks associated with mixing it with other substances, especially central nervous system depressants like alcohol or benzodiazepines. They should discuss any concerns or side effects with their healthcare provider. Patients undergoing treatment for opioid use disorder should adhere to the rules of their treatment program [2].

How is Methadone dispensed?


Methadone for pain management may be prescribed and dispensed like other prescription medications. However, methadone used for opioid treatment programs is typically dispensed through specially licensed opioid treatment programs (OTPs) or from a physician's office if they have the appropriate DEA registration and state licenses. Daily observed dosing is common in OTPs [2, 6].


**Sources:


1. "Methadone." *National Institute on Drug Abuse
, 14 June 2023, www.drugabuse.gov/publications/drugfacts/methadone.
2. "Methadone Side Effects, Uses, Dosage & Warnings." Drugs.com, www.drugs.com/methadone.html. Accessed 18 May 2024.
3. "Drug Patent Watch." DrugPatentWatch.com, www.drugpatentwatch.com.
4. "Pain Medications." National Institute of Neurological Disorders and Stroke, www.ninds.nih.gov/health-information/patient-care/treatment-vectors/pain-medications. Accessed 18 May 2024.
5. "Medication-Assisted Treatment (MAT)." Substance Abuse and Mental Health Services Administration, www.samhsa.gov/medication-assisted-treatment. Accessed 18 May 2024.
6. "DEA Diversion Control Division." Drug Enforcement Administration, www.deadiversion.usdoj.gov. Accessed 18 May 2024.



Other Questions About Methadone :

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AI-Drug Label Prescribing Information Alignment Report

28
28%
Grade D

Poor

Not Aligned

Patient Risk: Moderate

Summary

Substantial portions of the extracted claims are not supported by the provided FDA label text (multiple claims marked 'absent from the label'), including specific brand/manufacturer associations and multiple adverse-effect and safety claims (e.g., drowsiness, dizziness, nausea, vomiting, constipation, sweating, QT prolongation, 'take exactly as prescribed'). Several clinically important claims are therefore not reliably label-grounded.


Category Scores

Indication
75
Good
Dosage
55
Partial
Contraindications
60
Partial
Warnings
35
Poor
DrugInteractions
70
Good
SpecificPopulations
20
Poor
AdverseReactions
10
Poor
Administration
45
Partial

Accurate Statements

Methadone is a synthetic opioid agonist.
Mechanism of Action: "μ agonist; a synthetic opioid analgesic"
Methadone is used for moderate to severe pain not responsive to non-narcotic analgesics.
INDICATIONS AND USAGE: "For the treatment of moderate to severe pain..."
Methadone is used for detoxification and maintenance in opioid addiction (OTP context).
INDICATIONS AND USAGE: "temporary treatment of opioid dependence"; "detoxification or maintenance in opioid addiction"; outpatient maintenance/detoxification only by OTPs certified by SAMHSA and registered by DEA
Methadone has potential for abuse and is a Schedule II controlled substance.
DRUG ABUSE AND DEPENDENCE: "potential for being abused... is a Schedule II controlled substance"
Alcohol and other CNS depressants may produce additive CNS depression and should be avoided.
Information for Patients: "Alcohol and other CNS depressants may produce an additive CNS depression... and should be avoided."
Methadone requires cautious, highly individualized prescribing and particular vigilance during initiation/conversion/titration.
DOSAGE AND ADMINISTRATION: "cautious and highly individualized approach"; "Particular vigilance is necessary"
Methadone is associated with symptoms suggestive of arrhythmia (patients should seek immediate medical attention for palpitations/dizziness/lightheadedness/syncope).
Information for Patients: "symptoms suggestive of an arrhythmia (such as palpitations, dizziness, lightheadedness, or syncope)"
DEA registration applies to OTP provision of outpatient maintenance and detoxification.
INDICATIONS AND USAGE: "Outpatient maintenance and outpatient detoxification... may be provided only by ... OTPs ... registered by the Drug Enforcement Administration (DEA)"

Unsupported Statements

Methadone is available under several brand names, including Dolophine.
Not supported by the provided label text (marked 'absent from the label').
Methadone is marketed as Methadose.
Not supported by the provided label text (marked 'absent from the label').
Methadone binds to opioid receptors in the brain.
Label supports μ-agonism and CNS involvement but does not explicitly support the exact phrasing 'binds to opioid receptors in the brain' (marked 'partially supported' in evaluation notes; treated here as not exactly supported).
Methadone binding reduces feelings of pain.
Not supported by the provided label text (marked 'absent from the label').
Methadone can lessen cravings and withdrawal symptoms associated with opioid addiction.
No explicit 'cravings' statement supported by provided label citations (partially supported; cravings not explicitly supported).
Because methadone acts on opioid receptors, it can prevent or reduce the effects of illicit opioids.
Not supported by the provided label text (marked 'absent from the label').
Methadone is a long-established medication.
Not supported by the provided label text (marked 'absent from the label').
Original patents for methadone have long since expired, allowing for generic production.
Not supported by the provided label text (marked 'absent from the label').
The brand Dolophine has been associated with Roxane Laboratories.
Not supported by the provided label text (marked 'absent from the label').
The brand Dolophine has been associated with Hikma Pharmaceuticals.
Not supported by the provided label text (marked 'absent from the label').
Methadose has been manufactured by Mallinckrodt.
Not supported by the provided label text (marked 'absent from the label').
Common side effects of methadone include drowsiness.
Not supported by the provided label text (marked 'absent from the label').
Common side effects of methadone include dizziness.
Not supported by the provided label text (marked 'absent from the label').
Common side effects of methadone include nausea.
Not supported by the provided label text (marked 'absent from the label').
Common side effects of methadone include vomiting.
Not supported by the provided label text (marked 'absent from the label').
Common side effects of methadone include constipation.
Not supported by the provided label text (marked 'absent from the label').
Common side effects of methadone include sweating.
Not supported by the provided label text (marked 'absent from the label').
Methadone can cause QT prolongation.
Not supported by the provided label text (marked 'absent from the label').
Methadone is effective in treating opioid use disorder.
Label supports opioid dependence/addiction terminology; provided wording 'opioid use disorder' is not shown in the provided label text.
Patients prescribed methadone should take it exactly as prescribed.
Not supported by the provided label text (marked 'absent from the label').
Methadone for pain management may be prescribed and dispensed like other prescription medications.
Not supported by the provided label text (marked 'absent from the label').
Methadone used for OTPs may be dispensed from a physician's office if the physician has appropriate DEA registration and state licenses.
Not supported by the provided label text (marked 'absent from the label').
Daily observed dosing is common in OTPs.
Not supported by the provided label text (marked 'absent from the label').
Methadone has efficacy in managing chronic pain.
Not supported by the provided label text (marked 'absent from the label'); label provided only 'moderate to severe pain' not chronic-pain efficacy phrasing.
Studies have demonstrated methadone effectiveness in decreasing illicit opioid use.
Not supported by the provided label text (marked 'absent from the label').
Studies have demonstrated methadone effectiveness in lowering the risk of overdose among individuals with opioid use disorder.
Not supported by the provided label text (marked 'absent from the label').
Studies have demonstrated methadone effectiveness in lowering the risk of infectious disease transmission among individuals with opioid use disorder.
Not supported by the provided label text (marked 'absent from the label').

Contradictions

Low

AI Statement
Methadone can cause QT prolongation.

Label Reference
No QT/QTc or QT prolongation statement appears in provided label excerpts; therefore this is an unverified claim rather than a direct contradiction.

Low

AI Statement
Patients should take it exactly as prescribed.

Label Reference
No such instruction appears in provided label excerpts; therefore unverified rather than directly contradicted.


Important Omissions

Boxed warning status and specific boxed-warning text were not provided in the supplied label excerpts and thus cannot be assessed for alignment. The extracted claims set did not evaluate boxed-warning language.
Importance: High
Full adverse reactions list and severity/frequency details were not included in the provided label excerpts, yet multiple extracted claims asserted 'common side effects' (drowsiness/dizziness/nausea/vomiting/constipation/sweating).
Importance: High
Pediatric use, geriatrics, and other specific population warnings/adjustments beyond general caution were not addressed in extracted claims and cannot be fully evaluated against label sections for those populations.
Importance: Moderate

Safety Assessment

Potential Patient Risk: Moderate
Multiple statements in the extracted claims are not supported by the provided FDA label excerpts, including specific side-effect assertions and QT prolongation. Additionally, key label safety elements (boxed warning and full adverse reactions) were not available for verification in the provided excerpts, preventing confirmation that critical safety information was accurately conveyed.

Regulatory Assessment

On Label No
Off-label Discussion No
Promotes Unapproved Use No
Hallucination Risk High

Recommendation

Not Aligned

Primary Issue
Large proportion of extracted claims are not supported by the provided label text (many explicitly 'absent from the label'), including brand/manufacturer associations, specific 'common side effects,' QT prolongation, and instruction-specific claims.

Suggested Improvement
Restrict claims to statements explicitly present in the provided FDA label excerpts, remove unsupported brand/manufacturer and side-effect frequency assertions, and ensure any safety claims (e.g., QT/QTc, adverse reactions, boxed warnings) are supported by the actual label text.

Drug Brand Mention Assessment

Branding Score
68
Visibility
67
Mentioned
Ranking
#1
Sentiment
75
Recommendation Status
mentioned only
Brand Perception
Best Known For

a synthetic opioid agonist used to treat severe pain and opioid use disorder


Core Claims
  • Methadone is a synthetic opioid agonist used to treat severe pain and opioid use disorder.
  • Methadone binds to opioid receptors in the brain and reduces feelings of pain.
  • Methadone can lessen cravings and withdrawal symptoms associated with opioid addiction.
  • Common side effects include drowsiness, dizziness, nausea, vomiting, constipation, and sweating.
  • More serious risks include respiratory depression and cardiac arrhythmias, particularly QT prolongation.
Differentiators
  • Often used in maintenance therapy for opioid use disorder due to slow onset and long duration of action.
  • Because it acts on opioid receptors, it can prevent or reduce the effects of illicit opioids.

Pricing Perception: Not Mentioned
Competitors Mentioned
Company Visibility Sentiment Rank Recommended
Buprenorphine 38%
55 #10 No
Naltrexone 37%
55 #11 No
Methadone 0%
0 # No