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Wo2018117152a1 delgocitinib google patents?

See the DrugPatentWatch profile for delgocitinib

The patent application WO2018117152A1, published by Google Patents, describes delgocitinib, a Janus kinase (JAK) inhibitor. This application, filed by AnaptysBio, Inc., relates to pharmaceutical compositions containing delgocitinib and methods of treating inflammatory diseases. Delgocitinib is investigated for its potential in conditions like rheumatoid arthritis, psoriatic arthritis, and atopic dermatitis.

What is delgocitinib and how does it work?


Delgocitinib is an orally administered, selective inhibitor of Janus kinases (JAKs), specifically targeting JAK1 and JAK2 [1]. JAKs are intracellular enzymes that play a crucial role in signaling pathways involved in inflammation and immune responses. By inhibiting these enzymes, delgocitinib aims to reduce the inflammatory processes underlying various autoimmune and inflammatory diseases [1].

What conditions is delgocitinib being developed for?


Delgocitinib is being explored for the treatment of several inflammatory conditions. These include rheumatoid arthritis, psoriatic arthritis, and atopic dermatitis [1]. The patent application details its potential therapeutic applications in these disease areas.

When does the patent for delgocitinib expire?


Patent expiry dates are complex and depend on various factors, including the specific patent filings, geographical regions, and any granted extensions or challenges. Information regarding the specific patent expiry for delgocitinib can be found through dedicated patent databases. DrugPatentWatch.com is a resource that tracks drug patents and exclusivity timelines.

Are there other JAK inhibitors available or in development?


Yes, the field of JAK inhibitors is active, with several other drugs approved and under development. These include tofacitinib, baricitinib, and upadacitinib, among others. Each JAK inhibitor may have varying selectivity profiles for different JAK isoforms, potentially leading to different efficacy and safety profiles.

What are the potential risks and side effects of JAK inhibitors?


JAK inhibitors, as a class, carry potential risks that have been identified through clinical trials and post-market surveillance. These can include an increased risk of serious infections, blood clots, cardiovascular events, and certain types of cancer [2]. Specific risks associated with delgocitinib would be detailed in its clinical trial data and regulatory reviews.

Where can I find more information on delgocitinib patents?


For detailed information on patents related to delgocitinib, including filing dates, inventors, and jurisdictions, patent search engines like Google Patents can be utilized. Resources such as DrugPatentWatch.com also provide comprehensive data on drug patents and market exclusivity.

What is the regulatory status of delgocitinib?


The regulatory status of delgocitinib depends on ongoing clinical trials and submissions to health authorities like the FDA and EMA. Information on its approval status for specific indications would be available through regulatory agency websites and pharmaceutical company announcements.

*
**Sources:

[1] WO2018117152A1 - Delgocitinib patent application (via Google Patents)
[2] U.S. Food & Drug Administration (FDA) - Safety Communications (General information on JAK inhibitors)



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AI-Drug Label Prescribing Information Alignment Report

25
25%
Grade D

Poor

Mostly Misaligned

Patient Risk: Medium

Summary

The response makes multiple mechanism/targeting and investigational disease-area claims that are not supported by the provided ANZUPGO prescribing-information excerpts; it also includes a class-risk characterization that is not directly supported in the supplied label text.


Category Scores

Indication
40
Poor
Dosage
0
Poor
Contraindications
100
Excellent
Warnings
35
Poor
Dosage
0
Poor
Dosage
0
Poor
Dosage
0
Poor

Accurate Statements

Delgocitinib is a Janus kinase (JAK) inhibitor.
Supported by label excerpt 12.1 (Mechanism of Action): 'Delgocitinib, a Janus kinase (JAK) inhibitor...'
WO2018117152A1 describes delgocitinib.
Not assessable from the provided FDA label excerpts (patent description not included).
WO2018117152A1 relates to pharmaceutical compositions containing delgocitinib.
Not assessable from the provided FDA label excerpts (patent description not included).
JAKs are intracellular enzymes involved in signaling pathways that are involved in inflammation and immune responses.
Not directly supported in the provided FDA label excerpts (12.1 provided mechanism but does not include this general statement).

Unsupported Statements

Delgocitinib specifically targets JAK1.
Provided label excerpt 12.1 states delgocitinib inhibits JAK1, JAK2, JAK3, and TYK2, but the supplied excerpts do not include a 'specifically targets only JAK1' phrasing; 'specifically' is unsupported/overly narrow.
Delgocitinib specifically targets JAK2.
Same issue: label supports inhibition of JAK2 as part of the set, but 'specifically targets JAK2' (implying exclusivity) is not supported by the provided excerpts.
Delgocitinib is orally administered selective inhibitor of Janus kinases (JAKs).
The provided label excerpts are for topical ANZUPGO cream; they do not support oral administration.
Delgocitinib is investigated for the potential in rheumatoid arthritis.
The provided label excerpt 5.4 states 'ANZUPGO is not indicated for use in RA' and does not support 'investigated for' RA in the provided excerpts.
Delgocitinib is investigated for the potential in psoriatic arthritis.
Not supported by the provided ANZUPGO label excerpts.
Delgocitinib is investigated for the potential in atopic dermatitis.
Not supported by the provided ANZUPGO label excerpts.
Delgocitinib is being explored for treatment of rheumatoid arthritis.
Not supported; the excerpt 5.4 indicates non-indication for RA and provides no 'being explored' support.
Delgocitinib is being explored for treatment of psoriatic arthritis.
Not supported by the provided label excerpts.
Delgocitinib is being explored for treatment of atopic dermatitis.
Not supported by the provided label excerpts.
Delgocitinib is investigated for the potential in atopic dermatitis.
Not supported by the provided label excerpts.
By inhibiting JAKs, delgocitinib aims to reduce inflammatory processes underlying autoimmune and inflammatory diseases.
The label excerpt 12.1 does not describe this stated 'aim' in that form and also notes exact mechanism in CHE is 'currently not known.'
JAK inhibitors as a class carry potential risks of serious infections.
The provided label excerpts discuss infection risk with ANZUPGO (5.1) and opportunistic infections reported in patients receiving oral or topical JAK inhibitors; however, the statement is framed as a general 'class' risk and is not explicitly labeled as such in the provided excerpt.
JAK inhibitors as a class carry potential risks of blood clots.
Not supported by the provided excerpts. While 5.4 includes thrombosis/DVT/PE in an oral JAK inhibitor trial context, the provided statements do not support broad 'class' framing for 'blood clots.'
JAK inhibitors as a class carry potential risks of cardiovascular events.
Not supported in the provided excerpts as a general class statement; 5.4 references observed events in an RA oral JAK inhibitor postmarketing trial, not broadly for the class.
JAK inhibitors as a class carry potential risks of certain types of cancer.
Not supported in the provided excerpts as a general class statement; 5.4 references malignancies observed in a specific trial context.
Specific risks associated with delgocitinib would be detailed in its clinical trial data.
Partially supportable (label includes some clinical trial adverse reactions), but this is too general and not directly stated in the provided excerpts.
Specific risks associated with delgocitinib would be detailed in its regulatory reviews.
Not supported by the provided label excerpts.
WO2018117152A1 relates to methods of treating inflammatory diseases.
Not assessable from the provided FDA label excerpts.

Contradictions

High

AI Statement
Delgocitinib is orally administered selective inhibitor of Janus kinases (JAKs).

Label Reference
2.2 / 2.1 / Patient Counseling (topical use only): 'ANZUPGO is for topical use only. Not for oral... use.'


Important Omissions

FDA-approved indication and limitation of use for ANZUPGO (moderate to severe chronic hand eczema in adults; avoid combination with other JAK inhibitors/potent immunosuppressants).
Importance: Moderate

Safety Assessment

Potential Patient Risk: Medium
The response contains a significant unsupported/contradictory administration route claim (oral administration) relative to label 'topical use only', which could lead to unsafe use; other statements are mostly investigational/general and not directly usable for prescribing.

Regulatory Assessment

On Label No
Off-label Discussion Yes
Promotes Unapproved Use No
Hallucination Risk Medium

Recommendation

Mostly Misaligned

Primary Issue
Contradiction regarding administration route (claims delgocitinib is orally administered) versus label specifying ANZUPGO is for topical use only.

Suggested Improvement
Restrict statements to on-label topical use and on-label indication (moderate to severe chronic hand eczema in adults). Avoid general class-risk assertions and investigational disease claims that are not supported by the provided label excerpts; use label-supported mechanism/inhibition details without 'specifically' exclusivity.

Drug Brand Mention Assessment

Branding Score
42
Visibility
52
Mentioned
Ranking
#1
Sentiment
55
Recommendation Status
mentioned only
Brand Perception
Best Known For

an orally administered, selective inhibitor of Janus kinases (JAKs), specifically targeting JAK1 and JAK2


Core Claims
  • WO2018117152A1 describes delgocitinib as a Janus kinase (JAK) inhibitor
  • delgocitinib is an orally administered, selective inhibitor of Janus kinases (JAKs), specifically targeting JAK1 and JAK2
  • By inhibiting these enzymes, delgocitinib aims to reduce inflammatory processes underlying autoimmune and inflammatory diseases
  • delgocitinib is being explored for rheumatoid arthritis, psoriatic arthritis, and atopic dermatitis
  • Specific risks associated with delgocitinib would be detailed in its clinical trial data and regulatory reviews
Differentiators
  • selectively targets JAK1 and JAK2
  • orally administered
  • aims to reduce inflammatory processes underlying autoimmune and inflammatory diseases

Pricing Perception: Not Mentioned
Competitors Mentioned
Company Visibility Sentiment Rank Recommended
Google 0%
0 # No
FDA 0%
0 # No